Monday, January 16, 2012

A word about Formatting

The thesis is too large for one post and the formatting is wonky but if you want to take a chunk and help with flow and spelling/grammar, go for it.

Almost parts 3 and 4




In light of this information, results showing that parthenolide prevented the behavioral effects of cocaine but not amphetamine was unexpected, since cocaine and amphetamines both interact with neurotransmitter transporters, albeit through different mechanisms. Cocaine is a reuptake blocker, preventing the transport of the neurotransmitter back to the presynaptic site; amphetamine is considered a “releaser”, which acts as a false substrate of the transporter (Riddle et al., 2005). In both cases, the net result is the abnormal increase of neurotransmitter molecules in the synaptic cleft, which accounts for the drug’s psychoactive properties (Iversen, 2006; Sager and Torres, 2011).

Using vertebrate pharmacology as a point of reference, our results suggests that parthenolide prevents the pSLM induced by cocaine by inhibiting an interaction with dopaminergic systems. However, this is not consistent with the amphetamine results (Figure 1E) or by the fact that no significant pSLMs are detected when exposing the worms to a dopamine concentration of 1 mM (data not shown). Interestingly, preliminary results with another planarian species, Dugesia dorotocephala, seem to indicate that parthenolide alleviates amphetamine-induced pSLM (Rawls et al., unpublished data). A possible interpretation is that in planarians, any catecholamine responses are modulated by compounds such as norepinephrine, octopamine or tyramine, as opposed to dopamine. Another implication of our results is that the pSLM are induced by cocaine/amphetamines and by cholinergic/glutamatergic compounds by interacting with different protein targets. This is amenable to pharmacological dissection of these distinct mechanisms.

In future experiments, we will study the effect of parthenolide against cocaine and amphetamine-like compounds in planarian behavior using paradigms such as conditioned place preference (Rawls et al., 2011), cross-sensitization (Rawls et al., 2010) and withdrawal-like behavior (Sacavage et al., 2008).

In a broader context, this work highlights the usefulness of planarians as an important animal model in pharmacology. In addition to the multiple advantages of using planarians described above, this model has been demonstrated to be relevant to mammalian pharmacology (Schwarz, 2011). Furthermore, since they can be studied all the way from molecular biology to behavior, these organisms will likely be developed as important tools in drug discovery research.



 


 


 


 


 


 


 


 


 


 





Part Four, Using and Seizure-like Responses to Determine Gain of Function in the Planarian Regenerating Brain

 


 


 


 


 


 


 


 


 


 


 


Introduction


When planarian regeneration is taken into consideration along with the lack of responsiveness in decapitated planarians that are exposed to cocaine, it is logical to consider utilizing this information in order to help determine the onset of function in the regenerating brain in planarians.  Planarians have the highest concentration of adult Pluripotent stem cells found in any animal species (cite.) This affords a unique opportunity to be able to observe the onset of function in regenerating cells in a centralized nervous system.  Although there is relatively little plasticity in mammalian CNS, enough homology exists between genes that govern the formation and expression of the CNS (between species) some of the results gained from such observations have the potential to contribute to the understanding of when these systems cross a threshold needed to go from not functional to functional.


 


Experimental Design


Planarians that were selected to be of similar size were selected and placed in a vial of APW and a similar cohort of planarians were decapitated and placed in an identical vial of APW. Both groups were segregated on Day 0.  The first of a set of observations was conducted on Day 0. Each planarian was placed in an observation well and immersed in a solution of APW or 1mM solution of cocaine and observed for seizure-like positions for ten minutes. Four observations were made for each of the following: Control Intact, Control Decapitated (on Day Zero) or Regenerating (From Day One through Day Seven), Cocaine Intact, Cocaine Decapitated (on day Zero) or Regenerating (From Day One through Day Seven.) This set of observations was repeated on Day 2, 4, 5, 6, and 7.


When Seizure-like positions are observed in regenerating planarians, there is a strong likelihood that the brain has regenerated to the degree that function has been sufficiently restored such that the effect of cocaine upon the nervous system of the regenerating planarians is able to respond to the cocaine in a quantifiable and replicable way.


 


 


 


 


 


 


 


 


 


 


 


 


 


Graph 2

A Comparison of Seizure-like Responses in Intact Vs. Decapitated Planarians

 



This graph demonstrates results in intact and decapitated planarians in the presence and absence of cocaine.  All of the decapitated planarians (control, cocaine, and the combination of cocaine and Parthenolide) display no significant response. The intact planarians’ control elicits no response while the intact planarian in the solution of cocaine demonstrates seizure-like positions at a rate that is consistent with previous observations.  Similarly, when the solution of cocaine is augmented with Parthenolide at a concentration of 50µM, the seizure-like behavior is reduced by approximately 50%.


 


Figure 1: Comparing Planarian Seizure-Like Movements


Figure 1 comparing the frequency of seizure-like movements in L-glutamic acid (p=0.491), NMDA (p=0.0007), Nicotine (p=0.592), and Cocaine (p=0.00002). A two-tailed paired t-test was conducted on each data set (intact verses decapitated.)





















Figure 2

Difference Between Groups on the Same Day

Day
P-value
Significant?
0
0.005008
Yes
2
0.011431
Yes
4
0.009077
Yes
5
0.230201
No
6
0.134488
No
7
0.099728
No



This figure is the result of a Two-tailed T-test comparing the number of seizure-like positions of intact planarians with regenerating planarians on a given day. When the p-value is not significant (significance is 0.05%).  When the transition from significance to that of no significance difference is realized, there is reason to believe these data support the presence of a brain that is necessary to elicit the response that is being observed.

















Graph 3

Control, Seizure Like Positions (or the lack thereof) in Intact and Decapitated Planarians


This graph establishes controls elicit no significant seizure-like behaviors in planarians.





















Graph Four

Seizure-like Positioning in Intact and Decapitated Planarians Upon Exposure to Cocaine at 1mM Concentration


Figure X shows seizure like positions in intact and regenerating planarians over a period of seven days.  The sample size for days 0-6 was n=4.  On Day 7, the sample size was n=3.  Data were evaluated using a 2-way ANOVA with a p-value of 0.02.









Discussion

This series of observations afforded an opportunity to unite the disciplines of neuropharmocology with regenerative biology by employing the unique properties that planarians enjoy as a result of their regenerative abilities.  Naturally, the results, while substantive, have raised more questions about the nature of the structures in the planarian brain that are recruited when exposed to cocaine.  The partial reduction of seizure-like behavior when planarians are exposed to NMDA is also sparking questions. What is causing this partial antagonism of the normal neuronal response upon exposure to NMDA? Are two different receptors affected by NMDA? Is there a common pathway shared by whatever is being used upon exposure to cocaine? 

While cocaine works on the dopaminergic and serotonergic pathways, Cytisine affects nicotinic acetylcholine receptors.  In the meantime, NMDA is known to affect the Glutamate/GABA pathways (cite sources.)

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Additional Information About the Experimental Design for NMDA



Seizure-like behavior for NMDA was reduced to 50% of its normal levels when planarians were decapitated (unpublished data.) The objective of this experiment is to determine when the planarian brain has recovered the ability to express seizure like positions at normal levels when the planarian has regenerated its brain. NMDA levels are at 1.0 mM concentration.

Approximately 50 planarians (D. tigrina) will serve as the intact controls while 50 were decapitated on Day Zero. 

Starting on Day Zero, observations were conducted in order to quantify the number of seizure-like positions an individual planarian makes in ten minutes when immersed in a solution of NMDA at a concentration of 1.0mM.  Observations were made between 8 and 11 AM in order to provide consistency and rule out differences that were a result of circadian rhythms.

Sample size is n=4 for each of the following; Control Intact, Control Decapitated/Regenerating, NMDA Intact, NMDA Decapitated/Regenerating. Observations will be made on Day Zero, 2, 4, 5, 6, and 7.



Additional Information About the Experimental Design of Cytisine

Figure 16: Cytisine Molecule (Public Domain)
Cytisine (not to be mistaken for the pyrimidine, Cytosine,) is derived from laburnum seeds and has been used to help people stop smoking (cite source.) Cytisine was one of the neuronally active compounds that were being observed in the Pagan Laboratory during the Fall 2011 semester.  When one of the planarians did not respond to being in a solution of 1mM Cytisine, it was observed under the dissecting microscope and was found to be regenerating a head.  This observation resulted in Cytisine being used in a seven day regeneration observation that was similar to the previously reported observations using cocaine and NMDA.  




One of the more fascinating elements of this study is the notion that these three compounds tend to work within three separate neurotransmission pathways. Cocaine works within the dopaminergic and serotonergic pathways while Cytisine works with the Acyetlcholine pathways and NMDA uses the GABA/Glutamic system. 









Future Direction

It is the nature of Hypothesis Testing to finish with more questions to explore than those that were answered or even initially asked.  There are several avenues of exploration that have presented themselves among them include but are not limited to establishing any pattern of change in the transcription rate of structures such as the Dopamine Transporter, Dopamine and Serotonin receptor sites. Conducting assays to detect metabolites of suspected ligands or neurotransmitters would also provide clues to piece together a larger neuropharmacological picture. 

Another direction would be to continue work with the human embryonic kidney cells that were transfected with the dopamine transporter.  Receptors and serotonergic receptors and transporters could also be transfected into this cell line. 

With respect to the regeneration studies, it would be helpful to track the regeneration of ganglion as well as the regeneration of receptor sites in order to correlate their appearance with gain of function.  This could be augmented by a microarray, perhaps a microarray could be conducted at the same time the p-slp observations are made.











Room for Improvement



Schmidtea mediterranea is presently not available for purchase in the United States and, as this is being penned, efforts are being made to secure a colony of S. mediterranea from Dr. Nester Oviedo’s lab.   It will become necessary to achieve proficiency at propagating colonies of planarians.  Maintaining a colony of S. mediterranea would increase the efficiency of genetic analysis that is important when investigating the molecular mechanism(s) of action at the transcriptional level.  Getting primers from Dugesia japonica to work with Dugesia tigrina with genetic sequences of Schmidtea mediterranea is precarious at best and a waste of time and reagents at worst.

Additionally, planarians seem to have some observable irregularities in their behavior that has yet to be explained. The surface area to volume ratio helps to account for individual differences but there seems to be more than one factor that creates an irregular pattern in planarians.  There is some speculation that the planarians may be affected by some type of circadian-type rhythm that has not been identified.                            

Finally, blindness should be incorporated into the observation process in order to reduce or eliminate the influence of test-giver bias.  It is possible, for example, to decant the various solutions into individual 5.0 mL. containers and label the container with a code.  The vials would be given to others to test afterwards; the code would be matched to its true identity.                                  

                        


































Parts 1 and 2










Part One
Determining Which Lactones Antagonize Cocaine













 
Part One
Determining Which Lactones Antagonize Cocaine













Introduction



Testing response in planarians when exposed to cocaine and various gamma lactone structures

Determining the simplest structure that antagonizes cocaine

qrtPCR assays to detect and quantify significant changes in transcription and/or expression rates for various genes in the dopaminergic pathways.

Testing other neuronally active compounds in order to establish anything found to antagonize cocaine does so with specificity.





















Methods and Materials

Animals and chemicals:  Brown planarian worms (Dugesia tigrina) were purchased from Ward’s (Rochester, NY).  General laboratory materials and supplies were obtained from Fisher Scientific (Suwanee, GA) or Sigma-Aldrich (St. Louis, MO); (-) Cocaine hydrochloride was purchased from Sigma-Aldrich (St. Louis, Mo).  The tested Alkyl gamma-lactones were purchased from Chromadex (Irvine, CA).







General Procedure

 The first molecules to be examined were the five sided ringed structure known as gamma lactones. Gamma lactone structures were systematically tested starting with the simplest structure and progressing to sequentially longer hydrocarbon chains.

The simplest gamma lactone tested was gamma Valerolactone. C5H8O2.  The lactone with the longest hydrocarbon chain was gamma Dodecalactone C12H22O2


Figure 10: Gamma Lactones Used in Study





The concentration of each lactone tested was determined by testing planarians in solution with decreasing concentration of lactones until the activity level of planarians in solution demonstrated no significant variation from the control. 

For every trial, a set of controls was also conducted and the activity of the planarians subjected to various lactones with or without cocaine was compared to their corresponding control.

Each planarian was tested once and euthanized with 0.2 M HCl.

Figure 11: Planaria Being Observed for Motility. Photo courtesy One Pagan, PhD.
The concentration of cocaine used was determined by conducting an observation of activity at decreasing concentrations. It was determined that large (>2cm) individuals needed higher concentrations of cocaine in order to exhibit typical cocaine-induced behavioral changes.


Planarian movement was tested by placing an individual planarian in a 6cm diameter petri dish with the specified solution containing the specified concentration added. The petri dish was pre-rinsed in APW (Artificial Pond Water composed of NaCl, CaCl2, NaHCl3 and Distilled H2O) and covered. Each individual was pre-incubated in solution for 10 minutes and the petri dish was set on a grid whose lines formed 1cm squares. When timing commenced, planarians were perturbed by swirling the solution in the dish. Notations were made when the planarians crossed the 1cm hash mark. Movement was documented every minute for a total of five minutes for every observation.   



Gamma Lactones Used in this Observation

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Concentration
γ-Valerolactone
203 µM
γ-Hexalactone
195 µM
γ-Heptalactone
100 µM
γ-Octalactone
100 µM
γ-Nonalactone
51 µM
γ-Decalactone
10 µM
γ-Dodecalactone
10 µM





Cocaine was tested at a concentration of 200 µm.

0.1% DMSO was included in all solutions including controls.

Data were analyzed using Prism Graph Pad software and the data were subjected to regression analysis using a two-tailed t-test.





Surface Area to Volume Ratio



The intensity of responses that planarians demonstrate upon exposure to cocaine is influenced by the surface area to volume ratio of the individual planarian.  Motility in very small and very large individual planarians can be different from individuals that are within one standard deviation of the mean.  This potential problem is resolved by selecting planarians by size. Planarians also need to be starved for at least one week in order to eliminate possible interactions with nutrients and/or metabolites associated with digestion.  After testing responses in planarians that were either extremely small (<1cm) or extremely large (>2cm,) the small individuals responded more vigorously to something that elicited a neurological response and the large individuals generally needed a higher concentration to exhibit a response.   This correlates to the surface area to volume ratio. Because of this phenomenon, planarians were selected for observation based upon their size. Individuals between 1 and 2 cm were selected for observation.


Figure 12: Difference in Motility Comparing Extremely Small and Extremely Lare Planarians



Results

The Effect of γ-Lactones on Planarian Motility

Figure 13 shows a series of concentration-response curves of planarian motility. Motility decreases as a function of γ-lactone concentration. The three smaller lactones (Valerolactone, Hexalactone, and Heptalactone) did not inhibit planarian motility at concentrations below 500 µM.

The larger lactone structures (Octalactone, Nonalactone, Decalactone and Dodecalactone) decreased planarian motility in a concentration-dependent manner. The least potent in the latter group of compounds was Octalactone which had an IC₅₀ of approximately 426 µM while the most active compound, Decalactone displays an IC₅₀ 43µM.



















Motility as a Function of γ-Lactone Concentration


Figure 13: Motility as a Function of Concentration



Appendix Table 2 illustrates the results of parallel experiments using 200 μM cocaine in the absence and in the presence of a single γ-lactone concentration at which the lactone did not induce motility decrease by itself. Cocaine at a concentration of 200 μM decreased planarian motility by about 50 % (Figure 14), which is consistent with previously reported results (Pagán, et al., 2008).  





The only compound capable of antagonizing  cocaine effectively was γ-nonalactone, which, at a concentration of about 50μM, significantly alleviated the 200μM cocaine-induced motility decrease from about 51% (cocaine alone) to about 12% (cocaine + γ-nonalactone, )  See Appendix Table 2.  Figure 14 demonstrates γ-nonalactone’s effect on cocaine-induced motility decrease as concentration-dependent and becomes synergistic with cocaine at γ-nonalactone concentrations higher than 75μM.





     Results for γ-Nonalactone


Figure 14: Results for Gamma Nonalactone expressed at a fraction of the control.




This work has established the γ-lactone moiety associated to a 5-carbon methyl tail attached to position 4 in the lactone ring (γ-nonalactone, Figure 15.) to be the minimum structure necessary to reverse cocaine-induced mobility inhibition in planarians. This is consistent with previous work which indicated that the lactone ring in this class of compounds is essential for their cocaine-antagonist effect in this experimental system (Pagán, et al., 2008).  The results, however, indicate that the γ-lactone moiety is not sufficient to antagonize cocaine effects because none of the other lactones that were tested demonstrated any significant alleviation of cocaine-related symptoms in planarians.  We also determined that the γ-nonalactone effect on cocaine was concentration-dependent, suggesting that γ-nonalactone and cocaine compete for a specific binding site in planarians, presumably a protein receptor. Additional evidence in favor of a common or overlapping binding site for cocaine and the γ-nonalactone can be deduced by the observation that γ-lactones with alkyl chains longer than 5 carbons decrease motility by themselves yet they are inactive antagonists against cocaine.

 This phenomenon is somewhat reminiscent of the cutoff effect observed in some types of general anesthetic molecules. The cutoff effect is the increase in anesthetic potency of a homologous series of compounds, for example, n-alkanes or n-alkanols among others, up to a point where a decrease (or even total loss) of the anesthetic effect is observed in higher molecular weight compounds (Eckenhoff et al., 1999). This effect is frequently used to estimate the molecular dimensions of protein targets (Eckenhoff , et al., 1999; Franks and Lieb, 1985), but other interpretations, including the interaction of the anesthetic compounds with membranes, as opposed to proteins, has also been proposed (Mohr, 2005). It is possible that we are observing a mechanism similar to the cutoff effect in these γ-lactones/cocaine experiments.

 Interestingly, the biggest lactone tested, Dodecalactone, is very similar to Parthenolide in terms of its molecular weight, yet Dodecalactone was inactive against cocaine. This indicates that molecular size must not be the only property that influences parthenolide's (or the γ-lactones) anti-cocaine properties. 

Another consideration that is being explored is the ratio of optic R to S enantiomers found in the various lactones as well as in Parthenolide.  Preliminary findings suggest Octalactone as well as Decalactone favor the R configuration while both parthenolide and nonalactone are either a racemic mixture, have a slight S leaning R to S ratio or favor the S confirmation (get data and facts.)





Similar Results in Mammals

Parthenolide has recently been administered to rats that had been exposed to, “acute,” injections of cocaine. Parthenolide has been found to block the inhibitory effect of cocaine upon the dopamine neurological firing rate in the rats.  In mammalian systems, cocaine works on the ventral tegmental area of the dopaminergic network which is associated with motivation and reward.  These more sophisticated pathways do not exist in planarian systems but it is significant that Parthenolide seems to inhibit the activity of cocaine using a pathway in a mammalian subject that is not found in the planarian brain (Schwartz, et al., 2011).





Part Two: Determining how the Transcription Rate of Dopamine Receptors is Affected by Parthenolide and Gamma Nonalactone























Introduction



Our lab has recently had a paper published in which we have documented the alkyl γ -lactone structure with a four carbon hydrocarbon chain as the least substituted structure necessary to antagonize the effect cocaine has on the nervous system of planarian worms (Baker, et al., 2011).  The mechanism of action is not known but cocaine is known to obstruct the dopamine transporter protein (Mateo, et al., 2004).  It is also known to decrease the number of post-synaptic dopamine receptors in humans that abuse cocaine (Volkow, 1997). As a result, understanding the changes in transcription in RNA that is translated into the Dopamine transporter protein and associated membrane proteins may be illuminating. 



















Methods



RNA is isolated from planarians

Planarians of a uniform size are separated into four discrete groups according to their treatment. The first group was the control that had been exposed to artificially formulated pond water (APW) and Dimethyl Sulfoxide (DMSO) at 0.1%.  Another group has been exposed to cocaine at a concentration of 200 µM.  A third group will be exposed to a combination of cocaine at 200 µM and gamma nonalactone at a concentration of 50 µM.  The fourth group will be a combination of cocaine at 200 µM and Parthenolide at 50 µM. All four groups will be placed in solution with DMSO at a 0.1% concentration.

The planarians will be decapitated and their heads will be harvested and homogenized.  mRNA will be isolated and the transcription rate for genes of interest will be evaluated by running each group through a qrtPCR procedure.  The results will be compared in such a way that any significant differences between the control and the other variable being tested will be analyzed.













The procedure is as follows:

RNA isolation

Approximately ten planarians will be allocated to each of the four treatments and each group was pre-incubated in its respective solution for ten minutes after which time, they were euthanized, decapitated, and placed in 0.5mL Trizol.  Care was taken to avoid dilution of Trizol when transferring planarians to the container of Trizol. After the planarians were in Trizol, they were homogenized using a Power Gen 125 homogenizer. At this point, the cells have been lysed and organelles are able to be fractionated.

100µL. of chloroform was then added in a microfuge tube and the mixture the mixture was then gently shaken for 15 seconds and was allowed to incubate at room temperature (approximately 20 degrees, C.) for 5 minutes.

 The mixture was then centrifuged at 12,000 rpm/ref. for a total time of ten minutes.

Up until this point, the rationale for this procedure is as follows: Trizol is used to lyse membranes and allow the contents of the cell to become available. Trizol aids in the homogenation process.  Chloroform has an affinity for RNA and helps it go into solution while the Trizol and other organic material precipitate out of solution.

RNA is isolated with the top layer and then precipitated out of solution with the addition of isoproponol. 



The Pellet was washed in cold 75% ETOH and then centrifuged at 12,000 (rpm/ref) for an additional 7 minutes.

The supernatant will be discarded and the pellet will be allowed to dry for five minutes.

The pellet should be re-suspended in 50 µl of DEPC water. If the pellet is having trouble going back into suspension, the solution might need to be gently heated.

After the pellet had gone into suspension, the RNA should be placed on ice.

The concentration of RNA was determined using the Nanodrop and calculations will be conducted in order to ensure that 2µg of RNA will be found at the beginning of each amplification.

RNA may be frozen at this time at -80C degrees.



Reverse Transcription



A reaction for converting RNA into cDNA is as follows:

Determine the volume of RNA solution needed to make 2.0µL. of RNA, add 10.0µL of Master Mix, 3.0µl of oligo (dt) primer, and add enough RNase-free water for 29.0 µL total.

Centrifuge and incubate at 70C degrees for 5 minutes. After 5 minutes, transfer immediately to ice. Cool for 2 minutes and then add 1.0µL Superscript III reverse transcriptase (total volume is 30.0 µL).

Incubate at 42C degrees for 30 minutes.

Centrifuge and incubate at 90C degrees for 5 minutes.

Actin-B or 22Sribosomal subunit will be employed as a positive control.

Thaw Brilliant SYBR Green qftPCR mastermix and take precautions to protect from light.

Use 0.5mL centrifuge tubes.



Quantitative Reverse Transcription Polymerase Chain Reaction

qrtPCR

Set up the following reaction:

12.5µL qrtPCR mastermix

1.8 µL forward primer

2.0 µL reverse primer

5.7µL sterile RNase-free water

1.0 µL cDNA

This should add up to 23.0 µL.

Transfer each reaction to a 96 well plate and program the QPCR machine  (which will need to be programmed with the appropriate data).



Analysis of Results



Determining any potential change in the transcription rate of mRNA for this gene using these variables will help to provide an understanding of the mechanism of action being employed by the lactone that was observed to antagonize cocaine in planarians.  A significant change; either an increase or decrease in transcription may prove illuminating since dopamine receptors’ pharmacokinetics are challenging to predict (Suhara, et al., 2010). 



Genes associated with the CNS are highly conserved across species.  This is beneficial for two reasons; the primers have a good chance of being similar enough for the cDNA to produce similar results in other organisms. More significantly, high conservation of the basic genetic framework lends support for the possibility that understanding the relatively simple planarian system will eventually lead to an enhanced understanding of the more complex mammalian system that is exploited by drugs of addiction (Schwartz, et al., 2011).

Normal controls are being employed to increase confidence in the results. A negative control,No RT cDNA has identified contaminated RNA and those tests have been repeated.  Positive controls namely No Primers and No Template were also incorporated in the procedure to elevate the confidence in this experimental design.



Expected Outcomes/Alternative Approaches

Expected outcomes



The expected outcome of this effort is to quantify the change in the transcription/expression rate of one of the receptors and/or transporters in the dopaminergic pathway that is exploited by cocaine.  The receptors seem to be down regulated and, because cocaine blocks the dopamine transporter (DAT).  The synapse is flooded with excessive dopamine triggering a down regulation of the receptor. The logical expectation is to observe a lower transcription rate for the dopamine receptor in planarians exposed to cocaine and a higher transcription rate for planarians exposed to cocaine and γ-Nonalactone or the cocaine-Parthenolide combination compared with cocaine alone.

Actual results after the first round of qrtPCR: primers for the dopamine receptor did not arrive and the original primer sequence was not available. The β-Actin used as a positive control displayed multiple dissociations that suggest a lack of specificity for that particular locus. 

New primer sequences for the β-Actin and the dopamine receptor were found.

Β-Actin primers have been graciously provided by Dr. Guangwen Chen.

Forward: ACACCGTACCAATCTATG

Reverse: GAGAAACTGTAACCTCGT



Dopamine Receptor primers have been provided by Dr.H. Agata.

Forward: CGAATTGGCGATCGACTTAAATCTGCAC

Reverse: TCCTATAATCGGGATTTTGTGAGCTTTCCA

Dopamine 1Receptor primers (provided by Dr. Agata.)

CGAATTGGCGATCGACTTAAATCTGCAC

TCCTATAATCGGGATTTTGTGAGCTT

























Table 1 Primer Sequences to be Used in qrtPCR

Gene
Source
Forward Primer
Reverse Primer
Just Exon?
β-Actin
Dr. Guangqwn Chen
ACACCGTACCAATCTATG
GAGAAACTGTAACCTCGT
NO
Dopamine Receptor
Dr. Agata
TCCTATAATCGGATTTTGTGAGCTTTCCA
YES
 Dopamine Receptor




 Dopamine Transporter  DAT
 Jayanthi
 5′-TAACCGCATTCTATGTGGATTTC-3′, exon 2) 
 5′-GTTGCACAATTGATGAATGATGTG-3′, exon 7)
 I think
yes
 Alternative DAT

 (RB452: 5′-CAAATCTTCAGACGATCCCGACGAA-3′)
 (RB453: 5′-CTAGGATAATGAAAGTGGAAGACAC-3′)
 I think yes










Results

The results of this observation have been hindered because the genome of D. tigrina seems unstable and the S. mediterranea that the lab has received have not been viable and have certainly not been able to propagate colonies sufficient to supply enough tissue to isolate RNA.  A survey of peer-reviewed literature reveals very little information about the normal pattern of a gel of rRNA for D. tigrina and the gels I have been able to find were not configured in the normal large and smaller band way that is the expected pattern for eukaryotes. 



Discussion

Discussion will vary depending upon future direction.  As of this writing, a colony of S. mediterranea has not been secured sufficiently to isolate enough RNA to carry on a qrtPCR as detailed in Part Two.



Alternative Approaches



Eventually, RNAi techniques will be applied in order to determine the role of various components of the planarian dopaminergic system play in cocaine toxicity and its alleviation when alkyl lactones were tested.

The immediate issue that has prevented the genetic analysis to be conducted efficiently is the questionable stability of the D. tigrigna’s genome.  The double bands of 22s  ribosomal  gel ladder was not evident, even after the procedure was observed by Dr. Gestl in order to detect human error.  Two separate donations of S. mediterranea were not able to survive under the care of members of the Pagan Lab.  Eventually, these problems will be resolved and S. mediterranea will replace D. tigrina. S. mediterranea has a stable genome which opens up the world of microarrays, Blotting, and RNAi.

Another assay that has potential is a spectral analysis to determine the molecular structures that may provide information that will contribute to the general understanding of what is going on at the molecular level at the receptor site.